- Neostigmine
- Drug Class:
Acetylcholinesterase Inhibitor
- Category: Neurological
Disorders
- Pharmacological Family:
Peripheral Nervous System Agent
Neostigmine inhibits the
enzyme acetylcholinesterase, which breaks down acetylcholine
(a neurotransmitter that regulates muscle movement). This leads to an increased
and prolonged effect of acetylcholine, helping treat certain neuromuscular
disorders.
Contraindications:
- Hypersensitivity to neostigmine,
bromide, or any other component
- Gastrointestinal or urinary tract
obstruction
Side Effects:
- Headache
- Drowsiness
- Nausea and vomiting
- Abdominal cramps
- Increased urination
- Cold sweats
- Tingling or warmth in extremities
- Mild skin rash
Available
Forms:
- Injectable Solution: 0.5 mg/mL, 1
mg/mL
- Tablets: 15 mg